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YX-02-030M 是一种 PROTAC MDM2 降解剂。YX-02-030M 抑制 MDM2-p53 结合和 VHL-HIF1α 结合,IC50 分别为 63 nM 和 1.35 μM。YX-02-030M 结合 MDM2 并募集 VH
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