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SPP-002 是一种硫酸酯类似物,作为一种潜在的 Sialyltransferase (ST) 抑制剂。SPP-002 能够选择性地抑制 N-糖链唾液酸化,其抑制效力至少比未修饰的亲本胆酸 (LCA) 提高了一个数量级。SPP-002 通过
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