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NO-711 是一种新型强效、选择性 γ-氨基丁酸吸收抑制剂。NO-711 可抑制突触体 (IC50 = 47 nM)、神经元 (IC50 = 1238 nM) 和神经胶质细胞 (IC50 = 636 nM) 的 GABA 吸收(体外)。更多
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