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XL-281 (BMS-908662) 是口服有效的 RAF 激酶抑制剂,对 CRAF、B-RAF 和 B-RAFV600E 的 IC50 分别为 2.6、4.5 和 6 nM。XL-281 具有抗肿瘤活性。更多详情参考:https://ww
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