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I1421 是囊性纤维化跨膜传导调节器 (CFTR) 的激活剂,对 WT CFTR 电流的 EC50 为 64 nM。I1421 还可以变构激活多种导致囊性纤维化 (CF) 的突变体,具有较好的体内效力,其在小鼠中的口服生物利用度为 60%,
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SARS-CoV-2 3CLpro-IN-13 | MedChemExpress (MCE)
8CN | 2-氨基-3-氰基-4,5-环辛烷并噻吩 | MedChemExpress (MCE)
H1k | MedChemExpress (MCE)
1-[3’-O-[(4,4’-Dimethoxytriphenyl)methyl]-a-L-threofuranosyl]-N4-benzoylcytosine | MedChemExpress (MCE)
2',3'-Dideoxyuridine | MedChemExpress (MCE)
2-Amino-6-chloro-9-[(2,3,5-tri-O-benzoyl-2-C-Methyl-beta-D-ribofuranosyl)]-9H-purine | MedChemExpress (MCE)
2-Aminoadenosine | 2-氨基腺嘌呤核苷 | MedChemExpress (MCE)
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3’-O-Methyluridine | 3'-O-甲基尿苷 | MedChemExpress (MCE)