MCE 的所有产品仅用作科学研究或药证申报,我们不为任何个人用途提供产品和服务。
CAS No. : 86401-95-8
MCE 国际站:Methylprednisolone aceponate
产品活性:Methylprednisolone aceponate (ZK 91588) 是一种糖皮质激素和抗炎剂,具有较弱的全身副作用。Methylprednisolone aceponate 是一种选择性的糖皮质激素受体 (glucorticoid receptor) 配体。Methylprednisolone aceponate 可用于研究湿疹和其他炎症性皮肤病。
研究领域:Immunology/Inflammation | Vitamin D Related/Nuclear Receptor
作用靶点:Glucocorticoid Receptor
In Vitro: Methylprednisolone aceponate inhibits collagenase promoter activity (in HeLa cells), LPS-induced IL-12p40 secretion (in human PBMCs) and phytohemagglutinin-induced IFN-γ secretion (in human PBMCs) with IC50s of 9.3, 16.8, 15.2 nM.
Methylprednisolone aceponate induces MMTV promoter and TAT activities with EC50s of 21.8 and 20.5 nM respectively.
In Vivo: Methylprednisolone aceponate (topically applied, 50 μL,,Coroton oil-induced Evan blue edema) shows anti-inflammatory effect with an IC50 of 0.0015%, with low systemic side effect.
Methylprednisolone aceponate (0.0001%-0.1%, topically applied) inhibits oedema formation with ED50 of 0.002% in irritant contact dermatitis in mice and rat.
相关产品:Drug Repurposing Compound Library Plus | Clinical Compound Library Plus | Bioactive Compound Library Plus | Immunology/Inflammation Compound Library | Clinical Compound Library | Drug Repurposing Compound Library | Nuclear Receptor Compound Library | Non-steroidal Anti-Inflammatory Compound Library | Pain-Related Compound Library | Medroxyprogesterone acetate-d3 | Prednisolone acetate | Clobetasone butyrate | Mifepristone-13C,d3 | Deflazacort | C108297 | Nenocorilant | Methylprednisolone succinate | Medroxyprogesterone acetate | Betamethasone 21-phosphate-d5 | Betamethasone dipropionate-d10 | Fluticasone propionate-d5 | Methylprednisolone-d5 | Hydrocortisone (Standard) | Fluticasone furoate-d3 | Dexamethasone-d4 | Mizacorat | Beclometasone dipropionate | Ciclesonide (Standard) | Methylprednisolone-d2 | Beclometasone dipropionate-d10 | Prednisone-d8 | Prednisolone Tebutate | Hydrocortisone hemisuccinate | Betamethasone-d5-1 | OP-3633 | Glucocorticoid receptor agonist-1
热门产品线:重组蛋白 | 化合物库 | 天然产物 | 荧光染料 | PROTAC | 同位素标记物 | 寡核苷酸 | 抗体 | 点击化学
Trending products:Recombinant Proteins | Bioactive Screening Libraries | Natural Products | Fluorescent Dye | PROTAC | Isotope-Labeled Compounds | Oligonucleotides | Antibodies | Click Chemistry
品牌介绍:
• MCE (MedChemExpress) 拥有200 多种全球独家化合物库,我们致力于为全球科研客户提供前沿最全的高品质小分子活性化合物;
• 50,000 多种高选择性抑制剂、激动剂涉及各热门信号通路及疾病领;
• 产品种类涵盖各种重组蛋白,多肽,常用试剂盒 ,更有 PROTAC、ADC 等特色产品,广泛应用于新药研发、生命科学等科研项目;
• 提供虚拟筛选,离子通道筛选,代谢组学分析检测分析,药物筛选等专业技术服务;
• 设有专业的实验中心和严格的质控、验证体系;
• 提供 LC/MS、NMR、HPLC、手性分析、元素分析等各项质检报告,确保产品的高纯度、高品质;
• 产品的生物活性多经各国客户实验验证;
• Nature, Cell, Science 等多种顶级期刊及制药专利收录了MCE客户的科研成果;
• 专业团队跟踪最新的制药及生命科学研究进展,为您提供全球最新的活性化合物;
• 与世界各大制药公司及知名科研机构建立了长期的合作。