Norfluoxetine hydrochloride | MedChemExpress (MCE)
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Norfluoxetine hydrochloride
CAS No. : 57226-68-3
MCE 国际站:Norfluoxetine hydrochloride
产品活性:Norfluoxetine hydrochloride 是 Fluoxetine 的 N-去甲基化活性代谢物。Fluoxetine 是一种选择性血清素 (5-HT) 再摄取抑制剂,可通过细胞色素 P450 (CYP) 2D6、CYP2C19 和 CYP3A4 代谢为 Norfluoxetine hydrochloride。Norfluoxetine hydrochloride 抑制 5-HT 摄取并抑制 CaV3.3 T 电流 (IC50=5 μM)。Norfluoxetine hydrochloride 具有抗惊厥活性。
研究领域:GPCR/G Protein | Neuronal Signaling | Membrane Transporter/Ion Channel | Metabolic Enzyme/Protease
作用靶点:5-HT Receptor | Calcium Channel | Drug Metabolite
In Vivo: Pretreatment with Fluoxetine or Norfluoxetine hydrochloride (20mg/kg s.c.), as well as Phenytoin (30 mg/kg s.c.) and Clonazepam (0.1mg/kg s.c.) significantly increases both the rate and duration of survival, demonstrating a significant protective effect against Pentylenetetrazol-induced epilepsy.
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