中文名:RETRA
英文名:RETRA
英文别名:RETRA hydrochloride|RETRA|1036069-26-7|1173023-52-3|2-(4,5-dihydro-1,3-thiazol-2-ylsulfanyl)-1-(3,4-dihydroxyphenyl)ethanone;hydrochloride|2-[(4,5-Dihydro-2-thiazolyl)thio]-1-(3,4-dihydroxyphenyl)ethanonehydrochloride|Ethanone, 2-[(4,5-dihydro-2-thiazolyl
纯度:≥98%
货号:R344313
Cas号:1036069-26-7
存储温度:2-8°C储存
产品介绍:
它是p73的突变体p53依赖性激活剂,p53调控基因的激活剂和携带突变体p53的肿瘤细胞的抑制剂。大于50%的肿瘤表达突变体p53,该突变体的肿瘤抑制功能存在缺陷,并通过阻断p53家族成员p73促成恶性肿瘤。在人类癌症中p73的激活产生细胞毒性作用。RETRA可提高p73的表达水平,并从具有突变体53的抑制复合物中释放p73。然后在体内和体外产生抑癌作用。
查看阿拉丁官网此产品相关对应页面:https://www.aladdin-e.com/zh_cn/R344313.html
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