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URB-602;CAS:565460-15-3原装热销

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产品介绍

BML-EI348-0050 50 mg
BML-EI348-0010 10 mg

Selectively inhibits monoacylglycerol (MAG) lipase (IC50=28µM) via a noncompetitive mechanism. Does not inhibit FAAH, DAG lipase or COX-2. URB-602 selectively raises levels of 2-arachidonoylglycerol with no change in anandamide concentrationsin cells and tissues. In the same way anandamide levels were markely elevated by the FAAH inhibitor URB597 at 1µM.
Product Specification
Formula: C19H21NO2
MW: 295.4
Purity: ≥98% (TLC)
Appearance: Off-white solid.
CAS: 565460-15-3
Solubility: Soluble in DMSO (30mg/ml), 100% ethanol (10mg/ml) or dimethyl formamide (30mg/ml). also soluble in a 1:1 solution in DMSO:PBS, pH 7.2 (0.25mg/ml)
Long Term Storage: Ambient
Use/Stability: Store, as supplied, at room temperature for up to 1 year. Store solutions at -20°C for up to 3 months.
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途