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Cilostamide;CAS:68550-75-4原装订购

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BML-PD125-0025 25 mg
BML-PD125-0005 5 mg

Phosphodiesterase PDE3 inhibitor (IC50=5 nM). Blocks PKB/Akt signaling pathway by inhibition of Akt-activated PDE3B. Reverses the established effects of leptin on food intake and body weight. Blocks the leptin-induced tyrosine phosphorylation of STAT3 at the hypothalamic level.
Product Specification
Alternative Name: OCP 3689, OPS 3689, N-Cyclohexyl-N-methyl-4-(1,2-dihydro-2-oxo-6-quinolyloxy)butyramide
Formula: C20H26N2O3
MW: 342.2
Purity: ≥98% (TLC)
Appearance: White solid.
CAS: 68550-75-4
Solubility: Soluble in DMSO (25mg/ml).
Long Term Storage: Ambient
Use/Stability: Stable for at least 1 year after receipt when stored, as supplied, at room temperature. Stock solutions are stable for up to 3 months at -20°C.
Handling: Packaged under inert gas.
Protect from light and oxygen.
Long Term Storage: Ambient
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