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Ketanserin
| 品牌 | 厂商性质 | 产地 | 货期 |
|---|---|---|---|
| 阿拉丁 | 生产商 | 上海 | 现货 |
产品参数
| 货号 | CAS号 | 操作 |
|---|---|---|
| K129651-1g | 74050-98-9 | 询价 |
| K129651-250mg | 74050-98-9 | 询价 |
| K129651-50mg | 74050-98-9 | 询价 |
产品介绍
- 分子式 C22H22FN3O3
- 分子量395.43
- Beilstein号
- EC号
- MDL号 MFCD00083392
- PubChem编号
属性
| 熔点 | 228-232 °C |
| 溶解性 | Soluble in water (<1 mg/ml at 25 °C), DMSO (2 mg/ml at 25 °C), ethanol (<1 mg/ml at 25 °C), DMF (10 mg/ml), and methanol. |
| 存贮条件 | 储存温度-20°C |
描述
| 应用 | A selective serotonin antagonist. |
| 产品介绍 | Ketanserin 是一种特异性的5-HT2A 5-羟色胺受体拮抗剂，作用于大鼠和人5-HT2A，Ki为2.5 nM。 |
| 备注 | Ketanserin (Vulketan Gel) is specific 5-HT2A serotonin receptor antagonist with a Ki of 2.5 nM for rat and human 5-HT2A. |
| 生化机理 | Ketanserin is reported to have a high affinity for multiple G protein-coupled receptors, such as serotonin receptors. Ketanserin is a selective serotonin 5-HT2/5-HT1C antagonist. It has been used to distinguish between 5-HT1D and 5-HT1B receptor subtypes. Additional studies have noted that Ketanserin is able to differentiate between recombinant human forms of these receptors with a higher affinity for 5-HT1Dα receptors compared to 5-HT1Dβ receptors. |
| 别名 | 酮色林; 酮舍林; 凯坦色林; 凯他色林; 3-[2-[4-(4-氟苯甲酰)-1-哌啶基]乙基]-2,4[1H,3H]-喹唑二酮;R-49945;Perketan;R-49945;3-[2-[4-(4-Fluorobenzoyl)-1-piperidinyl]ethyl]-2,4(1H,3H)-quinazolinedione |
Ketanserin信息由上海阿拉丁生化科技股份有限公司为您提供，如您想了解更多关于Ketanserin报价、型号、参数等信息，欢迎来电或留言咨询。
注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途