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Formoterol Hemifumarate
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
阿拉丁 | 生产商 | 上海 | 现货 |
产品参数
货号 | CAS号 | 操作 |
---|---|---|
F129812-10mg | 43229-80-7 | 询价 |
F129812-50mg | 43229-80-7 | 询价 |
产品介绍
- 分子式 C19H24N2O4·1/2C4H4O4
- 分子量402.40
属性
溶解性 |
|
存贮条件 | 储存温度 2-8°C |
描述
应用 | A potent β2-AR agonist. |
产品介绍 | Formoterol Hemifumarate是一种有效的,选择性的,长效β2-肾上腺素受体激动剂,作用于β2和β1受体,pKd分别为8.12和5.58。 |
备注 | Formoterol hemifumarate is a potent, selective and long-acting β2-adrenoceptor agonist to β2 and β1 receptors with pKd of 8.12 and 5.58, respectively. |
生化机理 | Formoterol Fumarate is shown to be a potent β-AR adrenoceptor agonist, with a fast onset of effect on the isolated human bronchus model. This compound demonstrates a 330-fold selectivity for β2 over β1 receptors. Formoterol Fumarate has been reported to be 150-200 times more potent than isoprenaline. This agent has also been noted to reduce the loss of muscle mass in murine models. |
别名 | 富马酸福莫特罗; N-[2-羟基-5[(RS)-1-羟基-2-[(RS)-2-(4-甲氧基苯基)-1-甲基乙基胺]乙基]苯基]甲酰胺半富马酸;Foradil;N-[2-Hydroxy-5-[[(1RS)-1-hydroxy-2-[[(1RS)-2-(4-methoxyphenyl)-1-methylethyl]amino]ethyl]phenyl]formamide (E)-2-butenedioate |
Formoterol Hemifumarate信息由上海阿拉丁生化科技股份有限公司为您提供,如您想了解更多关于Formoterol Hemifumarate报价、型号、参数等信息,欢迎来电或留言咨询。
注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途