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细胞信号转导
ADL5859 HCl
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
阿拉丁 | 生产商 | 上海 | 现货 |
产品参数
货号 | CAS号 | 操作 |
---|---|---|
A127848-1mg | 850173-95-4 | 询价 |
A127848-10mg | 850173-95-4 | 询价 |
A127848-50mg | 850173-95-4 | 询价 |
A127848-5mg | 850173-95-4 | 询价 |
产品介绍
属性
溶解性 |
|
存贮条件 | 储存温度-20°C |
描述
应用 | A selective receptor agonist for the δ-opioid receptor |
产品介绍 | ADL5859是δ-阿片受体选择性激动剂,Ki为0.8 nM,对hERG有弱抑制性。 |
备注 | ADL5859 HCl is a δ-opioid receptor agonist with Ki of 0.8 nM, selectivity against opioid receptor κ, μ, and weak inhibitory activity at the hERG channel. Phase 2. |
生化机理 |
ADL-5859 (ADL5859) is an δ-opioid receptor agonist (Ki=0.84 nM, EC50=20 nM). ADL-5859 (ADL5859) is an agonist agent that selectively stimulates the δ-opioid receptor with potential application in a wide range of inflammatory, neuropathic and acute pain conditions. In addition, Delta agonists are thought to modulate other biological processes that may manifest themselves in disease states or conditions such as overactive bladder and depression.ADL-5859 (ADL5859) is useful for inflammatory, neuropathic and acute pain conditions. |
别名 | ADL5859; ADL 5859; N,N-二乙基-4-(5-羟基螺(2H-1-苯并吡喃-2,4'-哌啶)-4-基)苯甲酰胺盐酸盐;;ADL5859; ADL 5859;N,N-Diethyl-4-(5-hydroxyspiro[2H-1-benzopyran-2,4'-piperidin]-4-yl)benzamide hydrochloride; |
ADL5859 HCl信息由上海阿拉丁生化科技股份有限公司为您提供,如您想了解更多关于ADL5859 HCl报价、型号、参数等信息,欢迎来电或留言咨询。
注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途