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Minisite
细胞信号转导
BMS-927711
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
阿拉丁 | 生产商 | 上海 | 现货 |
产品参数
货号 | CAS号 | 操作 |
---|---|---|
B125641-10mg | 1289023-67-1 | 询价 |
B125641-25mg | 1289023-67-1 | 询价 |
B125641-100mg | 1289023-67-1 | 询价 |
产品介绍
- 分子式 C28H28F2N6O3
- 分子量534.56
属性
溶解性 | DMSO |
存贮条件 | 储存温度-20°C |
描述
生化机理 |
Calcitonin gene-related peptide (CGRP) is closely involved in the cascade of molecular events leading to migraine painful crisis. New CGRP-R antagonist, such as BMS-927711, is in the pipeline and its developments will outline the future of this drug class. BMS-927711 has good oral bioavailability in rat and cynomolgus monkey, attractive overall preclinical properties, and shows dose-dependent activity in a primate model of CGRP-induced facial blood flow. BMS-927711 is presently in phase II clinical trials. |
BMS-927711信息由上海阿拉丁生化科技股份有限公司为您提供,如您想了解更多关于BMS-927711报价、型号、参数等信息,欢迎来电或留言咨询。
注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途