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Pizotifen Malate
| 品牌 | 厂商性质 | 产地 | 货期 |
|---|---|---|---|
| 阿拉丁 | 生产商 | 上海 | 现货 |
产品参数
| 货号 | CAS号 | 操作 |
|---|---|---|
| P129438-500mg | 5189-11-7 | 询价 |
| P129438-100mg | 5189-11-7 | 询价 |
产品介绍
属性
| 熔点 | 365-366.8 °C |
| 溶解性 | Soluble in water (3 mg/ml), and DMSO (30 mg/ml). |
| 存贮条件 | 储存温度-20°C |
描述
| 应用 | An antagonist of muscarinic receptors. |
| 产品介绍 | Pizotifen Malate用于治疗用于经常性偏头痛。 |
| 备注 | Pizotifen Malate is a benzocycloheptane based agent used for recurrent migraine headaches. |
| 生化机理 | Pizotifen malate, a derivative of benzocycloheptathiophene, is a tricyclic compound found to be a potent inhibitor of SR-2 receptor activity. In addition, it has been found to display vasoconstrictor activity in vivo. Studies on mice suggest that Pizotifen malate may have embryotoxic effects due to decreased value of mitotic indices in bone marrow cells. Pizotifen malate has also been reported to have acute antagonistic affects on central muscarinic receptors. |
| 别名 | 苯噻啶苹果酸盐; 9,10-二氢-4-(1-甲基哌啶-4-亚基)-4H-苯并[4,5]环庚烷并[1,2-b]噻吩苹果酸盐 (1:1);Pizotyline malate; Pizotifan; BC105;9,10-Dihydro-4-(1-methylpiperidin-4-ylidene)-4H-benzo[4,5]cyclohepta[1,2-b]thiophene malate (1:1) |
Pizotifen Malate信息由上海阿拉丁生化科技股份有限公司为您提供，如您想了解更多关于Pizotifen Malate报价、型号、参数等信息，欢迎来电或留言咨询。
注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途