应用 |
Pomalidomide is a second generation immunomodulator, TNF-α inhibitor, and thalidomide analog. An inhibitor of LPS-induced TNFαrelease. |
产品介绍 |
Pomalidomide抑制LPS诱导的TNF-alpha释放, IC50为13 nM。 |
备注 |
Pomalidomide inhibits LPS-induced TNF-α release with IC50 of 13 nM. |
生化机理 |
Pomalidomide is tumor necrosis factor-α inhibitor and a new immunomodulator with an IC50 of 1 μM.Pomalidomide is thalidomide derivative that displays inhibition of LPS-induced TNFα release. Shows immunomodulator and anticancer effects. |
别名 |
CC-4047;3-氨基-N-(2,6-二氧代-3-哌啶基)邻苯二甲酰亚胺;泊马度胺;TNF-alpha抑制剂;IMiD 3;1,3-dioxo-2-(2,6-dioxopiperidin-3-yl)-4-aminoisoindoline;3-amino-N-(2,6-dioxo-3-piperidyl)phthalamide;4-Amino-2-(2,6-dioxo-3-piperidinyl)-1H-isoindole-1,3(2H)-dione |