Darifenacin HBr-分析测试百科网

Darifenacin HBr

面议

品牌：阿拉丁
厂商性质：生产商
产地类别：国产
产地：上海
货期：现货
服务地域：全国
规格：5
近期咨询：0

分子式 C28H30N2O2.HBr 分子量507.46 属性熔点 228-230 °C 敏感性对湿度敏感溶解性 Soluble in water (<1 mg/ml at 25 °C), chloroform, DMSO (1

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上海阿拉丁生化科技股份有限公司

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货号	CAS号	操作
D129992-5g	133099-07-7	询底价
D129992-250mg	133099-07-7	询底价
D129992-1g	133099-07-7	询底价
D129992-50mg	133099-07-7	询底价
D129992-10mg	133099-07-7	询底价

耗材描述

分子式 C₂₈H₃₀N₂O₂.HBr
分子量507.46

属性

熔点	228-230 °C
敏感性	对湿度敏感
溶解性	Soluble in water (<1 mg/ml at 25 °C), chloroform, DMSO (117 mg/ml at 25 °C), methanol, and ethanol (<1 mg/ml at 25 °C).
存贮条件	储存温度 2-8°C

描述

应用	An M3 muscarinic acetylcholine receptor blocker.
产品介绍	Darifenacin HBr是一种选择性的M3 muscarinic（M3蕈毒碱）受体拮抗剂，pKi为8.9。
备注	Darifenacin is a selective M3 muscarinic receptor antagonist with pK_i of 8.9.
生化机理	Darifenacin hydrobromide is an antispasmodic muscarinic antagonist, selective for blocking the M3 muscarinic acetylcholine receptor, which is primarily responsible for bladder muscle contractions. Darifenacin hydrobromide has 9 and 12-fold greater affinity for M3 compared to M1 and M5, respectively, and 59-fold greater affinity for M3 compared to both M2 and M4. Darifenacin is used clinically to treat urinary incontinence and overactive bladder syndrome.
别名	氢溴酸达非那新; {1-[2-(2,3-二氢苯并呋喃-5-基)乙基]-3-吡咯烷基}-2,2-二苯基乙酰胺氢溴酸盐;UK 88525-04;Enablex;Darifenacin hydrobromide;(3S)-1-[2-(2,3-Dihydro-5-benzofuranyl)ethyl]-α,α-diphenyl-3-pyrrolidineacetamide hydrobromide ;UK 88525-04;{1-[2-(2,3-Dihydrobenzofuran-5-yl)ethyl]-3-pyrrolidnyl}-2,2-diphenylacetamide hydrobromide;Diphenyl-acetamide hydrobromide

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