Mizolastine-分析测试百科网

Mizolastine

面议

品牌：阿拉丁
厂商性质：生产商
产地类别：国产
产地：上海
货期：现货
服务地域：全国
规格：3
近期咨询：0

分子式 C24H25FN6O 分子量432.49 Beilstein号 EC号 MDL号 PubChem编号属性溶解性 DMSO <1 mg/mL Water <1 mg/mL Ethanol <1 mg/mL 存贮条

上海阿拉丁生化科技股份有限公司

上海阿拉丁生化科技股份有限公司

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货号	CAS号	操作
M129245-1g	108612-45-9	询底价
M129245-200mg	108612-45-9	询底价
M129245-5g	108612-45-9	询底价

耗材描述

分子式 C₂₄H₂₅FN₆O
分子量432.49
Beilstein号
EC号
MDL号
PubChem编号

属性

溶解性	DMSO <1 mg/mL Water <1 mg/mL Ethanol <1 mg/mL
存贮条件	储存温度-20°C

描述

应用	Mizolastine是组胺H1受体拮抗剂，IC50为47 nM。
产品介绍	Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions. Target: Histamine H1-receptor Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions. It does not prevent the actual release of histamine from mast cells, just prevents it binding to receptors. Side effects can include dry mouth and throat. Mizolastine has demonstrated antiallergic effects in animals and healthy volunteers and anti-inflammatory activity in animal models. Double-blind trials have shown mizolastine to be significantly more effective than placebo and as effective as other second generation antihistamine agents, such as loratadine or cetirizine, in the management of patients with perennial or seasonal allergic rhinitis and in patients with chronic idiopathic urticaria. Available data also suggest that prophylactic administration of mizolastine is significantly more effective than placebo and as effective as prophylactic terfenadine in delaying the onset of symptoms of seasonal allergic rhinitis.
备注	Mizolastine is a histamine H1-receptor antagonist with IC50 of 47 nM used in the treatment of hay fever (seasonal allergic rhinitis), hives and other allergic reactions.
别名	咪唑司汀;SL 850324

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