应用 |
A multi-targeted inhibitor. |
产品介绍 |
Pazopanib HCl (GW786034 HCl)是一种新型的针对VEGFR-1, VEGFR-2, VEGFR-3, PDGFR, FGFR, c-Kit和c-fms等多个靶点的抑制剂,IC50分别是10 nM, 30 nM, 47 nM, 84 nM, 74 nM, 140 nM和146 nM。 |
备注 |
Pazopanib (GW786034) is a novel multi-target inhibitor of VEGFR1, VEGFR2, VEGFR3, PDGFR, FGFR, c-Kit and c-Fms with IC50 of 10 nM, 30 nM, 47 nM, 84 nM, 74 nM, 140 nM and 146 nM, respectively.Phase 2 |
生化机理 |
Pazopanib Hydrochloride (GW786034, Votrient, Armala) is a novel, multitargeted inhibitor of VEGFR-1, VEGFR-2, VEGFR-3, PDGFR, FGFR, c-Kit and c-fms with IC50 values of 10 nM, 30 nM, 47 nM, 84 nM, 74 nM, 140 nM and 146 nM, respectively. |
别名 |
GW786034;盐酸帕唑帕尼;GW786034; Votrient; Armala; GW 786034; GW-786034;Pazopanib hydrochloride |