P129722-1gPazopanib HCl (GW786034 HCl)
面议
- 阿拉丁
- 生产商
- P129722-1g
- 现货
- 全国
规格 |
---|
耗材描述
属性
溶解性 | Soluble in DMSO (17 mg/ml at 25 °C), water (<1 mg/ml at 25 °C), ethanol (<1 mg/ml at 25 °C), and 30% PEG400/0.5% Tween80/5% propylene glycol (30 mg/ml at 25 °C). |
存贮条件 | 储存温度-20°C |
描述
应用 | A multi-targeted inhibitor. |
产品介绍 | Pazopanib HCl (GW786034 HCl)是一种新型的针对VEGFR-1, VEGFR-2, VEGFR-3, PDGFR, FGFR, c-Kit和c-fms等多个靶点的抑制剂,IC50分别是10 nM, 30 nM, 47 nM, 84 nM, 74 nM, 140 nM和146 nM。 |
备注 | Pazopanib (GW786034) is a novel multi-target inhibitor of VEGFR1, VEGFR2, VEGFR3, PDGFR, FGFR, c-Kit and c-Fms with IC50 of 10 nM, 30 nM, 47 nM, 84 nM, 74 nM, 140 nM and 146 nM, respectively.Phase 2 |
生化机理 | Pazopanib Hydrochloride (GW786034, Votrient, Armala) is a novel, multitargeted inhibitor of VEGFR-1, VEGFR-2, VEGFR-3, PDGFR, FGFR, c-Kit and c-fms with IC50 values of 10 nM, 30 nM, 47 nM, 84 nM, 74 nM, 140 nM and 146 nM, respectively. |
别名 | GW786034;盐酸帕唑帕尼;GW786034; Votrient; Armala; GW 786034; GW-786034;Pazopanib hydrochloride |
猜你喜欢
感兴趣产品