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CAS No. : 2101958-02-3
MCE 国际站:Squarunkin A
产品活性:Squarunkin A 是一种有效的选择性 UNC119-内容物 (Cargo) 相互作用抑制剂,能够抑制 UNC119A 与肉豆蔻酰化的 Src N 末端肽相互作用 (IC50=10 nM)。Squarunkin A 会干扰细胞中 Src 激酶的活化。
研究领域:Protein Tyrosine Kinase/RTK
作用靶点:Src
In Vitro: Squarunkin A (2.5 μM, 0.625 μM, 0.078 μM, and 0.01 μM) treatment leads to a concentration-dependent reduction of Src phosphorylation.
Squarunkin A does not target the lipoprotein-binding sites of other lipoprotein chaperones, such as PDE6d, AIPL1, and RhoGDI, which bind S-prenylated proteins. Squarunkin A binds to UNC119 in cell lysate and interferes with Src activation.
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