耗材描述
Angiotensin II 5-valine
产品活性:Angiotensin II 5-valine 是血管紧张素受体 (angiotensin receptor) 的激动剂。
产品来源: https://www.medchemexpress.cn/Angiotensin-II-5-valine.html
研究领域:GPCR/G Protein
作用靶点:Angiotensin Receptor
In Vivo: By day 12, systolic blood pressure (SBP) increases significantly in Angiotensin II 5-valine infused rats (197±7 mm Hg).The development of hypertension in ANG II infused rats is prevented by losartan treatment. Blood and kidney samples are harvested, subjected to HPLC to separate Angiotensin II 5-valine (exogenous) from Ile5-ANG II (endogenous) and the fractions are measured by radioimmunoassay. In the Angiotensin II 5-valine infused rats treated with losartan, total plasma ANG II levels are elevated to a greater extent than in rats not treated with losartan (289±20 v 119±14 fmol/mL). However, losartan markedly decrease by 88% the enhancement of intrarenal Val5-ANG II content that occurred in the rats infused with Val5-ANG II alone.
相关产品:Bioactive Compound Library Plus | Peptidomimetic Library | Peptide Library | Angiotensin II human | Losartan | Telmisartan | Tranilast | Valsartan | A 779 | Buloxibutid | AVE 0991 | Irbesartan | Candesartan | Nitrosoglutathione | YS-49 | Olmesartan | Olodanrigan | PD 123319 ditrifluoroacetate | Sparsentan | Alamandine | Azilsartan medoxomil | CGP-42112 | Talfirastide acetate | TRV-120027 | Angiotensin III, human, mouse
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