耗材描述
Aviptadil
产品活性:Aviptadil 是一种血管活性肠多肽 (VIP) 类似物,具有强的血管舒张 (vasodilatory) 作用。Aviptadil 诱导肺血管扩张,抑制血管 SMCs 增殖、血小板聚集。Aviptadil 可用于肺纤维化、肺动脉高压 (PAH)、SARS-CoV-2 引起呼吸衰竭等的研究。
产品来源: https://www.medchemexpress.cn/Aviptadil.html
研究领域:Anti-infection
作用靶点:SARS-CoV
In Vivo: Aviptadil (500 μg/kg; Intravenous injection; Every other day; Three weeks) completely prevented and significantly reversed Monocrotaline (MCT) (HY-N0750) -induced Pulmonary Arterial Hypertension in Sprague Dawley rat models (PAH)). Aviptadil is synergistic with Bosentan (HY-A0013).
Aviptadil (150 μg/kg/d; Intraperitoneal pump; 2.5 μl/h; 4 weeks) can eliminate bronchial hyperreactivity (BHR) in Sprague-Dawley rats, with a characteristic of bronchiectasis.
Aviptadil (0.1, 3 μg/kg; Intravenous injection (i.v.)) can improve reperfusion injury in living rat lung transplantation models.
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