耗材描述
Nodakenin
产品活性:Nodakenin 是 Angelica decusiva 根中的主要香豆素苷。Nodakenin 抑制乙酰胆碱酯酶 (AChE) 活性,IC50 为 84.7 μM。
产品来源: https://www.medchemexpress.cn/nodakenin.html
研究领域:Neuronal Signaling
作用靶点:Cholinesterase (ChE)
来源:植物 | 唇形科 | 小叶铃子香 | 植物 | 伞形科
结构分类:苯丙素类 | 香豆素 | 结构分类
In Vitro: Nodakenin inhibits AChE activity in a dosedependent manner with an IC50 value of 84.7 μM.
In Vivo: Nodakenin (10 mg/kg, p.o.) reverses scopolamine-induced cognitive impairments in the passive avoidance test and the Y-maze test.Nodakenin (10 mg/kg, p.o.) reduces escape latency during training in the Morris water maze test.
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