耗材描述
DTP3
产品活性:DTP3 TFA 是一种有效的选择性 GADD45β/MKK7 抑制剂。DTP3 TFA 靶向 NF-κB 通路下游,具有抗癌活性。
产品来源: https://www.medchemexpress.cn/dtp3.html
研究领域:Cell Cycle/DNA Damage | JAK/STAT Signaling | Stem Cell/Wnt | Epigenetics | Protein Tyrosine Kinase/RTK
作用靶点:DNA/RNA Synthesis | JAK
In Vitro: DTP3 (10 μM; 1-21 days) causes the potent and tumor-selective induction of JNK activation and apoptosis.
In Vivo: DTP3 TFA (s.c.; 14.5 mg/kg/day; 28 days) has shown a dramatic shrinkage of the tumors, and virtually eradicates established subcutaneous myeloma xenografts in mice. ?
DTP3 TFA (intravenous injection; 10 mg/kg/day) has t1/2 of 1.26 hours, CL of 27.13 ML/min/kg, and Vd of 2.80 L/kg.
相关产品:Bioactive Compound Library Plus | Cell Cycle/DNA Damage Compound Library | Epigenetics Compound Library | Immunology/Inflammation Compound Library | JAK/STAT Compound Library | Kinase Inhibitor Library | NF-κB Signaling Compound Library | Protein Tyrosine Kinase Compound Library | Stem Cell Signaling Compound Library | Anti-Cancer Compound Library | Anti-Aging Compound Library | Differentiation Inducing Compound Library | Reprogramming Compound Library | Anti-Breast Cancer Compound Library | Anti-Lung Cancer Compound Library | Anti-Pancreatic Cancer Compound Library | Anti-Blood Cancer Compound Library | Anti-Obesity Compound Library | Targeted Diversity Library | Anti-Liver Cancer Compound Library | Peptide Library | Anti-Prostate Cancer Compound Library | Cancer Stem Cells Compound Library | Autoimmune Disease Compound Library | Highly Selective Inhibitors Library | Anti-Hematopathy Compound Library | Bioactive Compound Library Max | Cycloheximide | Actinomycin D | Oxaliplatin | Gemcitabine | Ruxolitinib | Bleomycin sulfate | Carboplatin | Mitomycin C | Cytarabine | 5-BrdU | Methotrexate | Streptozotocin | Tofacitinib | Anisomycin | Fludarabine | ART558 | Propidium Iodide | Deucravacitinib | Thymidine | Baricitinib | Upadacitinib | AG490 | Hydroxyurea | Daunorubicin hydrochloride | Fedratinib | Remdesivir | Capecitabine | Brequinar
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