应用 |
A selective and reversible inhibitor of fatty acid amide hydrolase (FAAH). |
产品介绍 |
JNJ-1661010是一种有效的,选择性的FAAH抑制剂,IC50分别为10 nM(大鼠)和12 nM (人类),作用于FAAH-1比作用于FAAH-2选择性高100倍以上。 |
备注 |
JNJ-1661010 is a potent and selective FAAH inhibitor with IC50 of 10 nM (rat) and 12 nM (human), exhibits >100-fold selectivity for FAAH-1 when compared to FAAH-2. |
生化机理 |
JNJ 1661010 is a selective and reversible inhibitor of fatty acid amide hydrolase (FAAH) (IC50 = 12nM). JNJ 1661010 can also cross the blood-brain barrier. |
别名 |
N-苯基-4-(3-苯基-1,2,4-噻二唑-5-基)-1-哌嗪甲酰胺;N-Phenyl-4-(3-phenyl-1,2,4-thiadiazol-5-yl)-1-piperazinecarboxamide |