耗材描述

• 分子式 C₁₉H₁₉N₅OS
• 分子量365.45

属性

熔点	240.48 °C
溶解性	Soluble in DMSO (36 mg/ml at 25 °C), water (<1 mg/ml at 25 °C), and ethanol (<1 mg/ml at 25 °C).
存贮条件	储存温度 2-8°C

描述

应用	A selective and reversible inhibitor of fatty acid amide hydrolase (FAAH).
产品介绍	JNJ-1661010是一种有效的，选择性的FAAH抑制剂，IC50分别为10 nM(大鼠)和12 nM (人类)，作用于FAAH-1比作用于FAAH-2选择性高100倍以上。
备注	JNJ-1661010 is a potent and selective FAAH inhibitor with IC50 of 10 nM (rat) and 12 nM (human), exhibits >100-fold selectivity for FAAH-1 when compared to FAAH-2.
生化机理	JNJ 1661010 is a selective and reversible inhibitor of fatty acid amide hydrolase (FAAH) (IC50 = 12nM). JNJ 1661010 can also cross the blood-brain barrier.
别名	N-苯基-4-(3-苯基-1,2,4-噻二唑-5-基)-1-哌嗪甲酰胺;N-Phenyl-4-(3-phenyl-1,2,4-thiadiazol-5-yl)-1-piperazinecarboxamide

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