Ranolazine dihydrochloride | 盐酸雷诺嗪 | MedChemExpress (MCE)
品牌 | 厂商性质 | 产地 | 货期 | 价格 |
---|---|---|---|---|
MedChemExpress (MCE) | 生产商 | 美国 | 现货 | 660 |
性能特点
Ranolazine dihydrochloride (CVT 303 dihydrochloride) 是一种抗心绞痛和抗缺血剂,可通过抑制内向钠电流的后期作用 (对 INa 和 IKr 的
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
10 mM * 1 mL | 95635-56-6 | ¥660.00 | 询底价 |
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Ranolazine dihydrochloride
CAS No. : 95635-56-6
MCE 国际站:Ranolazine dihydrochloride
产品活性:Ranolazine dihydrochloride (CVT 303 dihydrochloride) 是一种抗心绞痛和抗缺血剂,可通过抑制内向钠电流的后期作用 (对 INa 和 IKr 的 IC50 值分别为 6 μM 和 12 μM) 来发挥功效,而不会影响心率或血压。Ranolazine dihydrochloride 还是脂肪酸氧化的部分抑制剂。
研究领域:Membrane Transporter/Ion Channel | Neuronal Signaling | Autophagy
作用靶点:Calcium Channel | Sodium Channel | Autophagy
In Vivo: Ranolazine (Bolus injection 10 mg/kg and infusion 9.6 mg/kg/h; bolus injection; for 145 minutes; male Wistar rats) treatment significantly reduces infarct size and cardiac troponin T release in rats subjected to left anterior descending coronary artery occlusion-reperfusion.
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途