(S)-Amisulpride | (S)-氨磺必利 | MedChemExpress (MCE)
品牌 | 厂商性质 | 产地 | 货期 | 价格 |
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MedChemExpress (MCE) | 生产商 | 美国 | 现货 | 2585 |
性能特点
(S)-Amisulpride (Esamisulpride) 是一种有效的多巴胺 D2/D3 受体拮抗剂。(S)-Amisulpride 是 5-HT7 受体的拮抗剂,KI 值为 900 n
规格 | CAS号 | 价格 | 操作 |
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10 mM * 1 mL | 71675-92-8 | ¥2,585.00 | 询底价 |
(S)-Amisulpride 产品活性:(S)-Amisulpride (Esamisulpride) 是一种有效的多巴胺 D2/D3 受体拮抗剂。(S)-Amisulpride 是 5-HT7 受体的拮抗剂,KI 值为 900 nM。(S)-Amisulpride 具有抗精神和抗抑郁作用。 产品来源: https://www.medchemexpress.cn/s-amisulpride.html 研究领域:GPCR/G Protein | Neuronal Signaling 作用靶点:Dopamine Receptor | 5-HT Receptor In Vitro: (S)-Amisulpride (Esamisulpride) displays high affinity binding at both D2 and D3 receptors and is approximately twice as potent as racamisulpride and 20–50 times more potent than (R)-amisulpride at these receptors In Vivo: The (S)-amisulpride (10mg/kg, s.c.) stimulus is rapidly acquired and was shown to be dose-related, time dependent (effective between 30 and 120min) and stereoselective male C57BL/6 mice. 相关产品:Drug Repurposing Compound Library Plus | Clinical Compound Library Plus | Bioactive Compound Library Plus | GPCR/G Protein Compound Library | Neuronal Signaling Compound Library | Clinical Compound Library | Drug Repurposing Compound Library | Neurotransmitter Receptor Compound Library | Anti-Alzheimer's Disease Compound Library | Anti-Parkinson's Disease Compound Library | Neurodegenerative Disease-related Compound Library | Antidepressant Compound Library | 5-HT Receptor Compound Library | Coagulation and Anti-coagulation Compound Library | Heterocyclic Compound Library | Membrane Protein-targeted Compound Library | Membrane Receptor-targeted Compound Library | Dopamine Receptor Compound Library | Multi-Target Compound Library | Bioactive Compound Library Max | Clozapine N-oxide | MPTP hydrochloride | Oxidopamine hydrobromide | Chlorpromazine hydrochloride | L-DOPA | Serotonin hydrochloride | Dopamine hydrochloride | SCH-23390 hydrochloride | Harmine | Puerarin | Haloperidol | Pimozide | PNU-282987 | SKF 38393 hydrochloride | Scopolamine hydrobromide | Risperidone | Cabergoline | Vortioxetine | Olanzapine | Dihydroergotamine mesylate | Aripiprazole | Bromocriptine mesylate | GTS-21 dihydrochloride | Fluphenazine dihydrochloride 品牌介绍: MCE (MedChemExpress) 拥有数百种全球独家化合物,我们致力于为全球科研客户提供最新最全的高品质小分子活性化合物;10,000 多种高选择性抑制剂、激动剂涉及各热门信号通路及疾病领域;设有专业的实验中心和严格的质控、验证体系;提供 LC/MS、NMR、HPLC、手性分析、元素分析等各项质检报告,确保产品的高纯度、高品质;产品的生物活性多经各国客户实验验证;Nature, Cell, Science 等多种顶级期刊及制药专利收录了MCE客户的科研成果;专业团队跟踪最新的制药及生命科学研究进展,为您提供全球最新的活性化合物;与世界各大制药公司及知名科研机构建立了长期的合作。
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