化合物GR 103691 T11463

Product Introduction
Bioactivity


英文名: GR 103691

描述: GR 103691 是选择性的多巴胺 D3受体拮抗剂，Ki=0.4 nM。它对人多巴胺 D3的选择性超过 D4和 D1的 100 倍以上。

体外活性: GR 103691 显示出对α-1肾上腺素能受体（Ki: 12.6 nM）和5-羟色胺1A（5-HT1A）受体（Ki: 5.8 nM）的显著亲和力。

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 4.86 mg/mL (10 mM)


关键字: Inhibitor | GR-103691 | GR 103691 | GR103691 | Dopamine Receptor | inhibit

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途