化合物LSD1-IN-7 benzenesulfonate T11882

Product Introduction
Bioactivity


英文名: Pulrodemstat benzenesulfonate

描述: Pulrodemstat benzenesulfonate (CC-90011 benzenesulfonate) 是一种有效的口服活性赖氨酸特异性去甲基化酶 1 (LSD1) 抑制剂，IC50为 0.25 nM，具有抗癌活性。它诱导急性髓细胞性白血病和小细胞肺癌细胞分化，对 LSD2、MOA-A 和 MAO-B 的酶抑制作用较小。

体内活性: LSD1-IN-7 in combination with other LSD1 inhibitor can be treatment of cancer in a mammal, including breast cancer, lung cancer, prostate cancer, glioblastoma, or leukemia.

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 60 mg/mL(98.42 mM)


关键字: LSD1 | Pulrodemstat | oral | SCLC | reversible | CC-90011 | cell | CC90011 | anticancer | Histone Demethylase | differentiation | inhibit | Inhibitor | AML | Pulrodemstat benzenesulfonate | CC 90011

相关产品: GSK-J1 | JQKD82 | T-3775440 hydrochloride | Daminozide | CPI-455 HCl | Iadademstat dihydrochloride | QC6352 | KDM2B-IN-2 | Vafidemstat | LSD1-IN-25

相关库: Anti-Cancer Compound Library | Bioactive Compounds Library Max | Anti-Lung Cancer Compound Library | Inhibitor Library | Epigenetics Compound Library | Anti-Cancer Active Compound Library | Orally Active Compound Library | Methylation Compound Library | NO PAINS Compound Library | Bioactive Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途