化合物 T11964 T11964
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
50 mg | 1039825-68-7 | ¥13,800.00 | 询底价 |
25 mg | 1039825-68-7 | ¥10,600.00 | 询底价 |
100 mg | 1039825-68-7 | ¥17,500.00 | 询底价 |
Product Introduction
Bioactivity
英文名: MCH-1 antagonist 1
描述: MCH-1 antagonist 1 also inhibits CYP3A4 (IC50: 10μM).MCH-1 antagonist 1 is a potent melanin concentrating hormone (MCH-1) antagonist (Ki: 2.6 nM).
体外活性: MCH-1 antagonist 1 also inhibits cytochrome P450 3A4 (CYP3A4) (IC50:10 μM).
体内活性: Effect of MCH-1 antagonist 1 (dosed at 30 mg/kg, po) is measured on the body weight of DIO mice with the AUC0-6 h of 14760 h*ng/mL.MCH-1 antagonist 1 is administered to male C57BL/6J DIO mice to assess their pharmacokinetic profile.
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
关键字: MCH1 antagonist 1 | MCH 1 antagonist 1 | MCH-1 antagonist 1
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途