化合物 T12694 T12694
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
100 mg | 405940-76-3 | ¥19,500.00 | 询底价 |
50 mg | 405940-76-3 | ¥15,300.00 | 询底价 |
25 mg | 405940-76-3 | ¥11,700.00 | 询底价 |
Product Introduction
Bioactivity
英文名: Razaxaban hydrochloride
描述: Razaxaban hydrochloride is a highly potent, selective and orally active inhibitor of factor Xa(Ki of 0.19 nM),has strongly antithrombotic activity.
体外活性: Razaxaban shows good Caco-2 permeability. The anticoagulant activity of Razaxaban is evaluated in the in vitro human plasma activated partial thromboplastin time (aPTT) and human prothrombin time (PT) assays. Razaxaban shows a doubling of aPTT and PT at 6.1 μM and 2.1 μM, respectively. .
体内活性: Traetment with Razaxaban inhibits thrombus formation in a dose-dependent manner (ID50 of 1.6 μmol/kg/h in the rabbit arterio-venous shunt thrombosis model).
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
关键字: BMS561389 Hydrochloride | DPC906 Hydrochloride | DPC-906 Hydrochloride | Razaxaban hydrochloride | BMS 561389 Hydrochloride | Razaxaban Hydrochloride | BMS-561389 Hydrochloride | DPC 906 Hydrochloride
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途