化合物 T12945 T12945
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
25 mg | 1104662-66-9 | ¥10,600.00 | 询底价 |
100 mg | 1104662-66-9 | ¥17,500.00 | 询底价 |
1 mL | 1104662-66-9 | ¥4,970.00 | 询底价 |
5 mg | 1104662-66-9 | ¥3,730.00 | 询底价 |
50 mg | 1104662-66-9 | ¥13,800.00 | 询底价 |
2 mg | 1104662-66-9 | ¥3,190.00 | 询底价 |
Product Introduction
Bioactivity
英文名: SNT-207858 free base
描述: SNT-207858 free base is a selective, blood brain barrier penetrating, potent and orally active antagonist of melanocortin-4 (MC-4) receptor(IC50 of 22 nM (binding) and 11 nM (function), on the MC-4 receptor).
体外活性: SNT207858 binds to MC-4 receptor with an affinity of 22 nM, and shows a 170-fold selectivity vs. MC-3 and a 40-fold selectivity vs. MC-5.
体内活性: In mice,the tumor induced weight loss significantly reduced by SNT207858 (30 mg/kg; oral administration; once daily; 15 days).
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : 125 mg/mL (202.72 mM)
关键字: SNT-207858 free base | SNT207858 free base | SNT 207858 free base | SNT207858 | SNT 207858 | SNT-207858
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途