化合物ARP-100 T14322

Product Introduction
Bioactivity


英文名: ARP-100

描述: ARP-100 (MMP-2 Inhibitor III) 是选择性基质金属蛋白酶MMP-2抑制剂 (IC50=12 nM)。它对 MMP-1 (>50 μM)，MMP-3 (4.5 μM)，MMP-7 (>50 μM) 和MMP-9 (0.2 μM) 的抑制活性较小。它与 MMP-2 的 S1＇口袋相互作用，并在体外对基质胶的侵袭模型中显示抗侵袭特性。

体外活性: ARP-100 (50 nM) exhibits a significant reduction in the total number of invasive elongations[1].

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 96 mg/mL (263.43 mM)


关键字: metalloproteinase | Inhibitor | Matrix metalloproteinases | selective | matrigel | ARP 100 | matrix | invasion | anti-invasive | ARP100 | MMP | ARP-100 | inhibit

相关产品: JG26 | CGS 27023A | YH-306 | SB-3CT | Histatin 5 acetate | MMP13-IN-3 | Triolein | Morroniside | Doxycycline hydrochloride | Ethyl gallate

相关库: Angiogenesis related Compound Library | Bioactive Compounds Library Max | Inhibitor Library | Anti-Fibrosis Compound Library | Protease Inhibitor Library | NO PAINS Compound Library | Anti-Cardiovascular Disease Compound Library | Bioactive Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途