化合物CYM50308 T15032

Product Introduction
Bioactivity


英文名: CYM50308

描述: CYM50308 是选择性和高亲和力的鞘氨醇-1-磷酸受体 4 激动剂，EC50为 56 nM。它对 S1P4-R 的选择性比 S1P5-R 高 37 倍。

体外活性: CYM50308 shows low nanomolar S1P4-R agonist activity and exquisite selectivity over the other S1P-Rs subtypes. CYM50308 provides a valuable pharmacological tool to explore the effects of the S1P4-R signaling cascade and elucidate the molecular basis of the in vivo receptor function[1].

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 12 mg/mL (29.60 mM)


关键字: ML248 | LPL Receptor | CYM50308 | Lysophospholipid Receptor | selective | S1P4-R | ML-248 | CYM 50308 | receptor | Inhibitor | Potent | inhibit | CYM-50308 | ML 248

相关产品: Etrasimod | Phorbol 12-myristate 13-acetate | Ceranib-2 | K6PC-5 | PF-543 hydrochloride | Vibozilimod | SKI-178 | Fingolimod | GLPG2938 | W140 HBr

相关库: Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | GPCR Compound Library | Bioactive Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途