化合物ESI-05 T15247

Product Introduction
Bioactivity


英文名: ESI-05

描述: ESI-05 (NSC-116966) 是特异性的 cAMP 直接激活交换蛋白 2 (EPAC2) 拮抗剂(IC50:0.4 µM)，能够抑制 cAMP 诱导的 EPAC2 的活化，并 EAPC2 介导的 Rap1 的活化。

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 83.33 mg/mL (303.70 mM)


关键字: Diacylglycerol acyltransferase | diabetes | Inhibitor | inhibit | Intracranial hemorrhage (ICH) | Acyltransferase | cAMP | acyl-CoA:cholesterol acyltransferase | insulin secretion | mono- acylglycerol acyltransferase | NSC-116966 | exchange proteins directly activated by cAMP 2 (EPAC2) | neurological disorders | NSC116966 | ESI-05 | ESI 05 | ESI05 | GEF | Diglyceride acyltransferase

相关产品: KH7 | GLP-1R modulator L7-028 | Licoarylcoumarin | Methyl orsellinate | Panaxydol | CE3F4 | 0990CL | Citreorosein | Kushenol A | Trans-caffeic acid

相关库: Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | Inhibitor Library | GPCR Compound Library | Target-Focused Phenotypic Screening Library | NO PAINS Compound Library | Bioactive Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途