化合物 T15425 T15425

Product Introduction
Bioactivity


英文名: GSK1702934A

描述: GSK1702934A is a selective TRPC3 agonist. It modulates cardiac contractility and f arrhythmogenesis by activation of TRPC3.

体外活性: GSK1702934A causes a transient, non-selective conductance and prolonged action potentials in TRPC3-overexpressing myocytes but not in wild-type myocytes[2]. GSK1702934A is able to induce TRPC3/6-currents in HEK293 cells transduced with recombinant human TRPC3/6 (EC50 of 0.08 mM and 0.44 mM, respectively)[1]. GSK1702934A substantially promotes NCX currents in TRPC3-overexpressing myocytes[2].

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

关键字: GSK-1702934A | GSK1702934A

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途