化合物UNC0379 T1841

Product Introduction
Bioactivity


英文名: UNC0379

描述: UNC0379 是一种选择性的、底物竞争性的赖氨酸甲基转移酶 SETD8 抑制剂，IC50值为 7.3 μM，也选择性抑制其他 15 种甲基转移酶。

体外活性: UNC0379 与多肽底物存在竞争性作用，与辅酶SAM则表现出非竞争性作用。[1]

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 76 mg/mL (183.8 mM)
H2O : < 1 mg/mL (insoluble or slightly soluble)


关键字: UNC0379 | Histone Methyltransferase | UNC-0379 | neuroblastoma | lysine methyltransferase | pulmonary fibrosis | antitumor | UNC 0379 | Inhibitor | OVCAR3 | HGSOC | Ovarian cancer | inhibit | JHOS3

相关产品: CPI-169 racemate | HLCL-61 hydrochloride | SMYD3-IN-1 | OICR-9429 | MI-463 | Antitumor agent-101 | Valemetostat tosylate | UNC 0631 | CM-272 | EZH2-IN-15

相关库: Anti-Aging Compound Library | Anti-COVID-19 Compound Library | Bioactive Compounds Library Max | Inhibitor Library | Epigenetics Compound Library | Methylation Compound Library | Stem Cell Differentiation Compound Library | Histone Modification Compound Library | NO PAINS Compound Library | Chromatin Modification Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途