化合物BMY-14802盐酸盐 T22612
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
50 mg | 105565-55-7 | ¥3,630.00 | 询底价 |
10 mg | 105565-55-7 | ¥1,160.00 | 询底价 |
5 mg | 105565-55-7 | ¥726.00 | 询底价 |
25 mg | 105565-55-7 | ¥2,430.00 | 询底价 |
1 mg | 105565-55-7 | ¥288.00 | 询底价 |
500 mg | 105565-55-7 | ¥10,900.00 | 询底价 |
100 mg | 105565-55-7 | ¥5,230.00 | 询底价 |
Product Introduction
Bioactivity
英文名: BMY-14802 hydrochloride
描述: BMY-14802 hydrochloride (BMS 181100 hydrochloride) 是一种选择性的 σ 受体拮抗剂 (IC50 = 112 nM),具有抗精神病作用。 BMY-14802 hydrochloride 是 α1-肾上腺素能受体和 5-HT1A 的激动剂。
体外活性: BMY-14802 hydrochloride shows effects on the firing of 5-HTergic and catecholaminergic neurons and affects behaviors in a 5-HT1A-sensitive manner[3].
体内活性: Intraperitoneal administration of BMY-14802 hydrochloride (5-20 mg/kg) shows anti-dyskinetic efficacy across a 4-fold dose range against L-DOPA-induced dyskinesias without affecting the efficacy of L-DOPA against lesion-induced akinesia. BMY-14802 hydrochloride reduces D1 and D2 receptor agonist-induced dyskinesias[2].
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: H2O : 9.0 mg/mL (23.4 mM)
关键字: BMS 181100 Hydrochloride | BMS-181100 Hydrochloride | BMS181100 Hydrochloride | BMY14802 Hydrochloride | BMY 14802 Hydrochloride | BMY-14802 Hydrochloride
相关产品: Sigma-1 receptor antagonist 2 | BD1063 dhydrochloride | Sigma-1 receptor antagonist 3 | BMY-14802 | NE-100 hydrochloride | KSK67 | AD186 | Blonanserin | L-745870 trihydrochloride | Amitriptyline
相关库: Neurotransmitter Receptor Compound Library | Anti-Cancer Compound Library | Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | Neuronal Signaling Compound Library | GPCR Compound Library | Bioactive Compound Library
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途