化合物GX-674 T22829
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
5 mg | 1432913-36-4 | ¥7,000.00 | 询底价 |
100 mg | 1432913-36-4 | ¥17,500.00 | 询底价 |
50 mg | 1432913-36-4 | ¥13,800.00 | 询底价 |
Product Introduction
Bioactivity
英文名: GX-674
描述: GX-674 是一种具有高效和选择性的电压门控钠通道 1.7 (Nav1.7) 拮抗剂,在 -40 mV 时测得 IC50 值为 0.1 nM,可用于研究炎症和神经性疼痛。
体外活性: In HEK293 cells, the patch-clamp analysis was performed for human Nav channels. GX-674 shows a potent inhibition effect on Nav.1.7 (IC50= 0.1nM). GX-674 also displays substantial selectivity on different Nav subtypes. It shows much higher inhibitory effects on Nav 1.7 over other Nav isoforms, such as 100000 times more potent for Nav1.7 than for Nav 1.5. GX-74 is also reported to bind to a high-affinity, isoform-selective, and extracellularly accessible site on VSD4.[1]
存储条件: store at low temperaturePowder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : Soluble
关键字: GX 674 | GX674 | GX-674
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途