化合物FAUC-213 T24055

Product Introduction
Bioactivity


英文名: FAUC 213

描述: FAUC 213 是一种具有口服活性的‘、高度选择性的、可透过血脑屏障的多巴胺 D4受体完全拮抗剂，对 hD4.4的 Ki=2.2 nM。它对 D2和 D3受体的活性较低，对于 hD2、hD3的 Ki 分别为 3.4 μM、5.3 μM。它表现出非典型的抗精神病活性。

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 3.26 mg/mL (9.99 mM)


关键字: inhibit | p5-HT2 | orally | pα1 | BBB | AMPH | barrier | amphetamin | blood-brain | Inhibitor | FAUC 213 | Dopamine Receptor | p5-HT1 | antipsychotic

相关产品: U91356 | Flibanserin | Pipamperone | Metergoline | Nortriptyline hydrochloride | SCH-23390 hydrochloride | 9-FLUORENOL | Syrosingopine | Doxepin hydrochloride | Droperidol

相关库: Anti-Neurodegenerative Disease Compound Library | Neurotransmitter Receptor Compound Library | Anti-Parkinson's Disease Compound Library | Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | Neuronal Signaling Compound Library | Inhibitor Library | GPCR Compound Library | Orally Active Compound Library | Bioactive Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途