赖苯普利 T27827
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
1 mg | 109214-55-3 | ¥1,750.00 | 询底价 |
50 mg | 109214-55-3 | ¥12,600.00 | 询底价 |
100 mg | 109214-55-3 | ¥16,900.00 | 询底价 |
5 mg | 109214-55-3 | ¥4,360.00 | 询底价 |
10 mg | 109214-55-3 | ¥6,220.00 | 询底价 |
25 mg | 109214-55-3 | ¥9,390.00 | 询底价 |
Product Introduction
Bioactivity
英文名: Libenzapril
描述: Libenzapril (CGS 16617)是一种有效的血管紧张素转换酶抑制剂,可用于研究心肌损伤。
体内活性: The effect of intravenous (i.v.) libenzapril was studied in six healthy males by administering i.v. angiotensin I (AI) was administered in stepwise increments of 20 ng/kg/5 min until the subjects' systolic blood pressure (SBP) had increased 20-30 mm Hg above baseline. The mean baseline infusion of 63 ng/kg/5 min resulted in a significant (P < 0.05) increase in the ratio of AII to AI plasma levels from 0.52 +/- 0.46 to 7.92 +/- 4.48 and a SBP increase of 120 +/- 7.1 to 147 +/- 5.6. Within 15 minutes of starting the 1-mg infusion of libenzapril over 1.5 hours, the AII/AI ratio decreased to baseline values, and the SBP returned to baseline in 1 hour. Repeat AI challenges at 3.5 and 5 hours postdose did not increase SBP significantly. Even the 6.5-hour challenge demonstrated only a slight increase in SBP, with an AII/AI ratio of 0.26. At 24 hours, SBP was only 40% of the baseline response, demonstrating that libenzapril is a potent long-acting ACE inhibitor.[1]
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : < 1mg/ml (insoluble)
关键字: CGS-16617 | Libenzapril | CGS16617
相关产品: L-Isoleucyl-L-arginine | Rentiapril racemate | Garcinone B | Vicenin-1 | Ovotransferrin (328-332) | H-Ile-Pro-Pro-OH acetate | Tuna AI acetate | Temocaprilat | Isocrenatoside | Trandolapril
相关库: Bioactive Compounds Library Max | Inhibitor Library | Bioactive Compound Library
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途