化合物TUG891 T3433
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
500 mg | 1374516-07-0 | ¥10,900.00 | 询底价 |
5 mg | 1374516-07-0 | ¥728.00 | 询底价 |
50 mg | 1374516-07-0 | ¥3,590.00 | 询底价 |
2 mg | 1374516-07-0 | ¥398.00 | 询底价 |
1 mg | 1374516-07-0 | ¥282.00 | 询底价 |
25 mg | 1374516-07-0 | ¥2,420.00 | 询底价 |
10 mg | 1374516-07-0 | ¥1,180.00 | 询底价 |
1 mL | 1374516-07-0 | ¥732.00 | 询底价 |
100 mg | 1374516-07-0 | ¥5,190.00 | 询底价 |
Product Introduction
Bioactivity
英文名: TUG-891
描述: TUG-891 是一种选择性的长链游离脂肪酸受体 4 (FFA4/GPR120) 的激动剂。
激酶实验: Inhibition of recombinant human Mps1 by BAY 1161909 or BAY 1217389 is assessed in TRFRET-based in vitro kinase assays via phosphorylation of a biotinylated peptide (Biotin-Ahx-PWDPDDADITEILG-NH2). Under standard assay conditions kinase and test compound are preincubated for 15 min before enzyme reaction is started by addition of substrate and ATP upon 10 μM[1].
体外活性: TUG-891与LCFA α-亚麻酸在人体FFA4上显示出相似的信号特性,包括促进Ca2+动员、β-阿雷斯汀-1和β-阿雷斯汀-2的招募以及细胞外信号调节激酶的磷酸化。TUG-891激活人体FFA4还导致受体的快速磷酸化和内化[1]。
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
溶解度: DMSO : 36.4 mg/mL(100 mM)
H2O : < 1 mg/mL (insoluble or slightly soluble)
关键字: Inhibitor | inhibit | Free Fatty Acid Receptor | TUG-891 | FFAR
相关产品: RTI-13951-33 | Fevipiprant | GLPG1205 | Kisspeptin-10, human (TFA)(374675-21-5,FREE) | NE 52-QQ57 | GPR84 antagonist 8 | 4-CMTB | AMG 837 calcium hydrate | PW0787 | Questiomycin A
相关库: Membrane Protein-targeted Compound Library | Anti-Metabolism Disease Compound Library | Bioactive Compounds Library Max | Human Metabolite Library | Fluorochemical Library | GPCR Compound Library | Anti-Obesity Compound Library | Endocrinology-Hormone Compound Library | Target-Focused Phenotypic Screening Library | Bioactive Compound Library
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途