HA-100 hydrochloride T38842
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
25 mg | 141543-63-7 | ¥10,600.00 | 询底价 |
Product Introduction
Bioactivity
英文名: HA-100 hydrochloride
描述: HA-100 hydrochloride is a powerful protein kinase inhibitor, exhibiting IC50 values of 4 μM, 8 μM, 12 μM, and 240 μM for cGMP-dependent protein kinase (PKG), cAMP-dependent protein kinase (PKA), protein kinase C (PKC), and MLC-kinase, respectively. Additionally, HA-100 hydrochloride is utilized as a ROCK inhibitor.
体外活性: HA-100 hydrochloride inhibits MLC-kinase and PKC competitively with respect to ATP, with K i s of 61 and 6.5 μM, respectively[1].
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
关键字: HA-100 Hydrochloride | HA100 hydrochloride | HA100 Hydrochloride | HA 100 hydrochloride | HA 100 Hydrochloride
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途