冬绿苷 T3S0509

Product Introduction
Bioactivity


英文名: Gaultherin

描述: Gaultherin 是一种分离自 Gaultheria yunnanensis 中的天然水杨酸酯衍生物。它是一种非甾体类抗炎药，具有止痛和抗炎作用，与 Aspirin 相比没有胃溃疡作用。

体外活性: The synthesis of Gaultherin (1) and its analogs was carried out to provide 11 glycosides under phase-transfer catalytic conditions. METHODS AND RESULTS: The activities of all synthesized compounds were evaluated by nitric oxide production inhibitory assay in vitro. Methyl 2-O-(4-O-β-d-galactopyranosyl)-β-d-glucopyranosylbenzoate (5f) showed significantly anti-nociceptive and anti-inflammatory effects by the evaluation in vivo. Structure-activity relationships within these compounds were discussed.

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 50 mg/mL (112.01 mM)


关键字: salicylate | NSAID | Gaultheria | yunnanensis | Gaultherin | Inhibitor | analgesic | anti-inflammatory | inhibit | non-steroidal

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相关库: Anti-Aging Compound Library | Anti-Cancer Compound Library | Mitochondria-Targeted Compound Library | Selected Plant-Sourced Compound Library | Bioactive Compounds Library Max | Neuronal Signaling Compound Library | Natural Product Library for HTS | Miao medicine Compound Library | Natural Product Library | Bioactive Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途