化合物S 38093 HCl T4087

Product Introduction
Bioactivity


英文名: S 38093 HCl

描述: S 38093 HCl 是一种新型的脑渗透性 H3 受体拮抗剂/反向激动剂。

激酶实验: PI3K inhibition by LY294002 is determined in a radiometric assay using purified, recombinant enzymes with 1 μM ATP. The kinase reaction is carried out for 1 hour at room temperature (24oC) and is terminated by addition of PBS. IC50 values are subsequently determined using a sigmoidal dose-response curve fit (variable slope). CK2 and GSK3β (glycogen synthase kinase 3β) inhibition are established by kinase selectivity screening. LY294002 is tested against the Upstate panel of kinases in 10 μM ATP.[4]

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: DMSO : 25 mg/mL (76.96 mM)


关键字: S 38093 HCl

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