化合物VU 0364439 T6160

Product Introduction
Bioactivity


英文名: VU 0364439

描述: VU 0364439是一种mGlu4阳性变构调节剂，EC50为19.8 nM。

体内活性: VU 0364439 由于其药代动力学性质不理想，限制了其作为体内工具的应用。相比于RLM（剩余2%），该化合物在HLM中表现出更好的稳定性（剩余63%）。[1]

存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year

溶解度: H2O : < 1 mg/mL (insoluble or slightly soluble)
Ethanol : < 1 mg/mL (insoluble or slightly soluble)
DMSO : 79 mg/mL (187.1 mM)


关键字: Metabotropic glutamate receptors | VU-0364439 | VU0364439 | Inhibitor | mGluR | VU 0364439 | inhibit

相关产品: (S)-3,4-DCPG HCl | Foliglurax | CBiPES hydrochloride | TCN238 | (S)-ATPO | mGluR3 modulator-1 | LYPLAL1-IN-1 | LSN2463359 | TAT-GluA2 3Y acetate(1404188-93-7 free base) | IEM 1754 2HBr

相关库: Anti-Neurodegenerative Disease Compound Library | Neurotransmitter Receptor Compound Library | Glutamine Metabolism Compound Library | Membrane Protein-targeted Compound Library | Bioactive Compounds Library Max | Neuronal Signaling Compound Library | Target-Focused Phenotypic Screening Library | NO PAINS Compound Library | Bioactive Compound Library

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注：该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案，不可用于临床诊断或治疗等相关用途