化合物 Encequidar, HCl T68568
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
50 mg | 849675-88-3 | ¥13,800.00 | 询底价 |
100 mg | 849675-88-3 | ¥17,500.00 | 询底价 |
25 mg | 849675-88-3 | ¥10,600.00 | 询底价 |
Product Introduction
Bioactivity
英文名: Encequidar, HCl
描述: Encequidar, also known as HM-30181, is an oral P-glycoprotein (P-gp) inhibitor developed to enhance the oral bioavailability of P-gp substrate drugs. Encequidar showed the highest potency (IC(50)=0.63nM) among several MDR1 inhibitors, including cycloporin A, XR9576, and GF120918, and effectively blocked transepithelial transport of paclitaxel in MDCK monolayers (IC(50)=35.4nM). Encequidar is currently under clinical trials.
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
关键字: Encequidar hydrochloride | Encequidar, HCl | HM30181 | HM-30181 | HM 30181
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途