化合物 SIM010603 T71576
品牌 | 厂商性质 | 产地 | 货期 |
---|---|---|---|
TargetMol | 生产商 | 美国 | 现货 |
性能特点
生化试剂,可用于动物细胞实验
规格 | CAS号 | 价格 | 操作 |
---|---|---|---|
50 mg | 1032265-67-0 | ¥16,800.00 | 询底价 |
100 mg | 1032265-67-0 | ¥21,500.00 | 询底价 |
25 mg | 1032265-67-0 | ¥12,800.00 | 询底价 |
Product Introduction
Bioactivity
英文名: SIM010603
描述: SIM010603 is a structurally novel, oral, multi-targeted receptor tyrosine kinase inhibitor. SIM010603 inhibited stem cell factor receptor (Kit), vascular endothelial growth factor receptor-2 (VEGFR-2), platelet-derived growth factor receptor-β (PDGFR-β), glial cell line-derived neurotrophic factor receptor (Rearranged during Transfection; RET), and Fms-like tyrosine kinase-3 (FLT3) with IC(50) values between 5.0 and 68.1 nmol/l. SIM010603 inhibited the phosphorylation of PDGFR-β and VEGFR-2. Moreover, SIM010603 inhibited endothelial cell proliferation, endothelial cells chemotaxis, and corneal angiogenesis.
存储条件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year
关键字: SIM-010603 | N-Desmethyl-4-hydroxytamoxifen | Z-Endoxifen HCl | SIM010603 | SIM 010603 | 4-Hydroxy-N-desmethyltamoxifen | Endoxifen hydrochloride
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注:该产品未在中华人民共和国食品药品监督管理部门申请医疗器械注册和备案,不可用于临床诊断或治疗等相关用途